http://purl.uniprot.org/citations/15012983 | http://www.w3.org/1999/02/22-rdf-syntax-ns#type | http://purl.uniprot.org/core/Journal_Citation |
http://purl.uniprot.org/citations/15012983 | http://www.w3.org/1999/02/22-rdf-syntax-ns#type | http://purl.uniprot.org/core/Journal_Citation |
http://purl.uniprot.org/citations/15012983 | http://www.w3.org/2000/01/rdf-schema#comment | "Substituted 3-amino-2-hydroxyamides and related hydroxyamides and acylhydrazines were identified as inhibitors of human methionine aminopeptidase-2 (MetAP2). Examination of substituents through parallel synthesis and iterative structure-based design allowed the identification of potent inhibitors with good selectivity against MetAP1. Diacylhydrazine 3t (A-357300) was identified as an analogue displaying inhibition of methionine processing and cellular proliferation in human microvascular endothelial cells (HMVEC)."xsd:string |
http://purl.uniprot.org/citations/15012983 | http://purl.org/dc/terms/identifier | "doi:10.1016/j.bmcl.2003.12.031"xsd:string |
http://purl.uniprot.org/citations/15012983 | http://purl.org/dc/terms/identifier | "doi:10.1016/j.bmcl.2003.12.031"xsd:string |
http://purl.uniprot.org/citations/15012983 | http://purl.uniprot.org/core/author | "Kim K.H."xsd:string |
http://purl.uniprot.org/citations/15012983 | http://purl.uniprot.org/core/author | "Kim K.H."xsd:string |
http://purl.uniprot.org/citations/15012983 | http://purl.uniprot.org/core/author | "Park C."xsd:string |
http://purl.uniprot.org/citations/15012983 | http://purl.uniprot.org/core/author | "Park C."xsd:string |
http://purl.uniprot.org/citations/15012983 | http://purl.uniprot.org/core/author | "Wang J."xsd:string |
http://purl.uniprot.org/citations/15012983 | http://purl.uniprot.org/core/author | "Wang J."xsd:string |
http://purl.uniprot.org/citations/15012983 | http://purl.uniprot.org/core/author | "Yang F."xsd:string |
http://purl.uniprot.org/citations/15012983 | http://purl.uniprot.org/core/author | "Yang F."xsd:string |
http://purl.uniprot.org/citations/15012983 | http://purl.uniprot.org/core/author | "Kawai M."xsd:string |
http://purl.uniprot.org/citations/15012983 | http://purl.uniprot.org/core/author | "Kawai M."xsd:string |
http://purl.uniprot.org/citations/15012983 | http://purl.uniprot.org/core/author | "Patel J."xsd:string |
http://purl.uniprot.org/citations/15012983 | http://purl.uniprot.org/core/author | "Patel J."xsd:string |
http://purl.uniprot.org/citations/15012983 | http://purl.uniprot.org/core/author | "Craig R.A."xsd:string |
http://purl.uniprot.org/citations/15012983 | http://purl.uniprot.org/core/author | "Craig R.A."xsd:string |
http://purl.uniprot.org/citations/15012983 | http://purl.uniprot.org/core/author | "Sheppard G.S."xsd:string |
http://purl.uniprot.org/citations/15012983 | http://purl.uniprot.org/core/author | "Sheppard G.S."xsd:string |
http://purl.uniprot.org/citations/15012983 | http://purl.uniprot.org/core/author | "Henkin J."xsd:string |
http://purl.uniprot.org/citations/15012983 | http://purl.uniprot.org/core/author | "Henkin J."xsd:string |
http://purl.uniprot.org/citations/15012983 | http://purl.uniprot.org/core/author | "Lesniewski R."xsd:string |
http://purl.uniprot.org/citations/15012983 | http://purl.uniprot.org/core/author | "Lesniewski R."xsd:string |