| http://purl.uniprot.org/citations/27749053 | http://www.w3.org/1999/02/22-rdf-syntax-ns#type | http://purl.uniprot.org/core/Journal_Citation |
| http://purl.uniprot.org/citations/27749053 | http://www.w3.org/2000/01/rdf-schema#comment | "Previously disclosed TAFIa inhibitors having a urea zinc-binding motif were used as the starting point for the development of a novel class of highly potent inhibitors having a sulfamide zinc-binding motif. High-resolution X-ray cocrystal structures were used to optimize the structures and reveal a highly unusual sulfamide configuration. A selected sulfamide was profiled in vitro and in vivo and displayed a promising ADMET profile."xsd:string |
| http://purl.uniprot.org/citations/27749053 | http://purl.org/dc/terms/identifier | "doi:10.1021/acs.jmedchem.6b01276"xsd:string |
| http://purl.uniprot.org/citations/27749053 | http://purl.uniprot.org/core/author | "Schreuder H.A."xsd:string |
| http://purl.uniprot.org/citations/27749053 | http://purl.uniprot.org/core/author | "Kohlmann M."xsd:string |
| http://purl.uniprot.org/citations/27749053 | http://purl.uniprot.org/core/author | "Czech J."xsd:string |
| http://purl.uniprot.org/citations/27749053 | http://purl.uniprot.org/core/author | "Evers A."xsd:string |
| http://purl.uniprot.org/citations/27749053 | http://purl.uniprot.org/core/author | "Halland N."xsd:string |
| http://purl.uniprot.org/citations/27749053 | http://purl.uniprot.org/core/author | "Czechtizky W."xsd:string |
| http://purl.uniprot.org/citations/27749053 | http://purl.uniprot.org/core/author | "Follmann M."xsd:string |
| http://purl.uniprot.org/citations/27749053 | http://purl.uniprot.org/core/author | "Kallus C."xsd:string |
| http://purl.uniprot.org/citations/27749053 | http://purl.uniprot.org/core/date | "2016"xsd:gYear |
| http://purl.uniprot.org/citations/27749053 | http://purl.uniprot.org/core/name | "J Med Chem"xsd:string |
| http://purl.uniprot.org/citations/27749053 | http://purl.uniprot.org/core/pages | "9567-9573"xsd:string |
| http://purl.uniprot.org/citations/27749053 | http://purl.uniprot.org/core/title | "Sulfamide as Zinc Binding Motif in Small Molecule Inhibitors of Activated Thrombin Activatable Fibrinolysis Inhibitor (TAFIa)."xsd:string |
| http://purl.uniprot.org/citations/27749053 | http://purl.uniprot.org/core/volume | "59"xsd:string |
| http://purl.uniprot.org/citations/27749053 | http://www.w3.org/2004/02/skos/core#exactMatch | http://purl.uniprot.org/pubmed/27749053 |
| http://purl.uniprot.org/citations/27749053 | http://xmlns.com/foaf/0.1/primaryTopicOf | https://pubmed.ncbi.nlm.nih.gov/27749053 |
| http://purl.uniprot.org/uniprot/#_P09955-mappedCitation-27749053 | http://www.w3.org/1999/02/22-rdf-syntax-ns#object | http://purl.uniprot.org/citations/27749053 |
| http://purl.uniprot.org/uniprot/P09955 | http://purl.uniprot.org/core/mappedCitation | http://purl.uniprot.org/citations/27749053 |